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Bioorganic Chemistry
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Volume 92, November 2019, Hidden issue
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1. Editorial Board
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2. Issue TOC
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3. Discovery of certain benzyl/phenethyl thiazolidinone-indole hybrids as potential anti-proliferative agents: Synthesis, molecular modeling and tubulin polymerization inhibition study
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Dilep Kumar Sigalapalli, Venkatesh Pooladanda, Priti Singh, Manasa Kadagathur, ... Nagendra Babu Bathini.
4. New A2A adenosine receptor antagonists: a structure-based upside-down interaction in the receptor cavity
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Catia Lambertucci, Andrea Spinaci, Michela Buccioni, Diego Dal Ben, ... Rosaria Volpini.
5. Dual VEGFR-2/PIM-1 kinase inhibition towards surmounting the resistance to antiangiogenic agents via hybrid pyridine and thienopyridine-based scaffolds: Design, synthesis and biological evaluation
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Tác giả
Ola H. Rizk, Mohamed Teleb, Marwa M. Abu-Serie, Omaima G. Shaaban.
6. Novel conjugates with dual suppression of glutathione S-transferases and tryptophan-2,3-dioxygenase activities for improving hepatocellular carcinoma therapy
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Tác giả
Shixian Hua, Xinyi Wang, Feihong Chen, Shaohua Gou.
7. Novel N-benzylpyridinium moiety linked to arylisoxazole derivatives as selective butyrylcholinesterase inhibitors: Synthesis, biological evaluation, and docking study
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Tác giả
Fahimeh Vafadarnejad, Elahe Karimpour-Razkenari, Bilqees Sameem, Mina Saeedi, ... Tahmineh Akbarzadeh.
8. Synthesis, biological activity and molecular modeling of a new series of condensed 1,2,4-triazoles
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Tác giả
Youness El Bakri, Ilias Marmouzi, Meryem El Jemli, El Hassane Anouar, ... El Mokhtar Essassi.
9. Germacrane-type sesquiterpenoids with cytotoxic activity from Sigesbeckia orientalis
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Tác giả
Na Liu, Cong Wu, Jin-hai Yu, Kong-kai Zhu, ... Hua Zhang.
10. Vernodalidimer L, a sesquiterpene lactone dimer from Vernonia extensa and anti-tumor effects of vernodalin, vernolepin, and vernolide on HepG2 liver cancer cells
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Tác giả
Sanit Thongnest, Pornsuda Chawengrum, Siriporn Keeratichamroen, Kriengsak Lirdprapamongkol, ... Somsak Ruchirawat.
11. Chemical constituents from Lonicera japonica flower buds and their anti-hepatoma and anti-HBV activities
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Lanlan Ge, Lingyun Xiao, Haoqiang Wan, Jiemei Li, ... Xiaobin Zeng.
12. Biflavones from Ginkgo biloba as inhibitors of human thrombin
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Tian-Ran Chen, Ling-Hua Wei, Xiao-Qing Guan, Chao Huang, ... Wen-Zhi Guo.
13. Ultrasound mediated efficient synthesis of new 4-oxoquinazolin-3(4H)-yl)furan-2-carboxamides as potent tyrosinase inhibitors: Mechanistic approach through chemoinformatics and molecular docking studies
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Nilam C. Dige, Prasad G. Mahajan, Hussain Raza, Mubashir Hassan, ... Sung-Yum Seo.
14. Nusbiarylins, a new class of antimicrobial agents: Rational design of bacterial transcription inhibitors targeting the interaction between the NusB and NusE proteins
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Yangyi Qiu, Shu Ting Chan, Lin Lin, Tsun Lam Shek, ... Cong Ma.
15. Novel 3,4-dihydro-4-oxoquinazoline-based acetohydrazides: Design, synthesis and evaluation of antitumor cytotoxicity and caspase activation activity
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Le Cong Huan, Phuong-Thao Tran, Cao Viet Phuong, Phan Huy Duc, ... Nguyen-Hai Nam.
16. Biscoumarin-1,2,3-triazole hybrids as novel anti-diabetic agents: Design, synthesis, in vitro α-glucosidase inhibition, kinetic, and docking studies
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Mohammad Sadegh Asgari, Maryam Mohammadi-Khanaposhtani, Mitra Kiani, Parviz Rashidi Ranjbar, ... Mir Hamed Hajimiri.
17. Discovery of HWL-088: A highly potent FFA1/GPR40 agonist bearing a phenoxyacetic acid scaffold
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Zheng Li, Qiang Ren, Xuekun Wang, Zongtao Zhou, ... Qianqian Qiu.
18. Spirocyclic sulfonamides with carbonic anhydrase inhibitory and anti-neuropathic pain activity
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Y. Kalisha Vali, Rambabu Gundla, Om V. Singh, Yasinalli Tamboli, ... Claudiu T. Supuran.
19. Design and synthesis of fluorogenic substrate-based probes for detecting Cathepsin B activity
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Shusheng Wang, Brady G. Vigliarolo, Morshed A. Chowdhury, Jennifer N.K. Nyarko, ... Christopher P. Phenix.
20. Synthesis and biological evaluation of a novel series of curcumin-peptide derivatives as PepT1-mediated transport drugs
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Jiyun Zhang, Hongmei Wen, Fei Shen, Xinzhi Wang, ... Wei Li.
21. Physapubescin I from husk tomato suppresses SW1990 cancer cell growth by targeting kidney-type glutaminase
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Kai-Yin Yang, Can-Rong Wu, Meng-Zhu Zheng, Ruo-Tian Tang, ... Hua Li.
22. A dual-emission fluorescent probe for discriminating cysteine from homocysteine and glutathione in living cells and zebrafish models
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Zhengliang Lu, Yanan Lu, Xin Sun, Chunhua Fan, ... Liying Gao.
23. Discovery of indoline derivatives that inhibit esophageal squamous cell carcinoma growth by Noxa mediated apoptosis
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Dong-Jun Fu, Miaomiao Li, Sai-Yang Zhang, Jiang-Feng Li, ... Tao Hu.
24. Pyrazole[3,4-d]pyridazine derivatives: Molecular docking and explore of acetylcholinesterase and carbonic anhydrase enzymes inhibitors as anticholinergics potentials
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Parham Taslimi, Fikret Türkan, Adnan Cetin, Hakan Burhan, ... Fatih Şen.
25. Coumarin tethered cyclic imides as efficacious glucose uptake agents and investigation of hit candidate to probe its binding mechanism with human serum albumin
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Dinesh S. Reddy, Manasa Kongot, Vishal Singh, Neha Maurya, ... Amit Kumar.
26. Synthesis of d-desthiobiotin-AI-2 as a novel chemical probe for autoinducer-2 quorum sensing receptors
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Vanessa Miranda, Inês M. Torcato, Karina B. Xavier, M. Rita Ventura.
27. The application of safe for humans and the environment Polyversum antifungal agent containing living cells of Pythium oligandrum for biotransformation of prochiral ketones
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Renata Kołodziejska, Renata Studzińska, Agnieszka Tafelska-Kaczmarek, Hanna Pawluk, ... Alina Woźniak.
28. Synthesis, in-vitro cholinesterase inhibition, in-vivo anticonvulsant activity and in-silico exploration of N-(4-methylpyridin-2-yl)thiophene-2-carboxamide analogs
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Gulraiz Ahmad, Nasir Rasool, Komal Rizwan, Imran Imran, ... Umer Rashid.
29. Synthesis, anticancer activity and molecular docking studies on 1,2-diarylbenzimidazole analogues as anti-tubulin agents
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Ya-Liang Zhang, Rong Yang, Lin-Ying Xia, Ruo-Jun Man, ... Hai-Liang Zhu.
30. Design, synthesis, and molecular docking study of new piperazine derivative as potential antimicrobial agents
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Mahadev Patil, Anurag Noonikara Poyil, Shrinivas D. Joshi, Shivaputra A. Patil, ... Alejandro Bugarin.
31. Design, synthesis and molecular docking of benzophenone conjugated with oxadiazole sulphur bridge pyrazole pharmacophores as anti inflammatory and analgesic agents
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Zabiulla, A.R. Gulnaz, Yasser Hussein Eissa Mohammed, Shaukath Ara Khanum.
32. Synthesis and comparative carbonic anhydrase inhibition of new Schiff’s bases incorporating benzenesulfonamide, methanesulfonamide, and methylsulfonylbenzene scaffolds
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Adel S. El-Azab, Alaa A.-M. Abdel-Aziz, Silvia Bua, Alessio Nocentini, ... Claudiu T. Supuran.
33. Xanthones from the stems of Cudrania tricuspidata and their inhibitory effects on pancreatic lipase and fat accumulation
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Yang Hee Jo, Seon Beom Kim, Jong Hoon Ahn, Ayman Turk, ... Mi Kyeong Lee.
34. Design and evaluation of non-carboxylate 5-arylidene-2-thioxo-4-imidazolidinones as novel non-competitive inhibitors of protein tyrosine phosphatase 1B
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Rosaria Ottanà, Paolo Paoli, Giulia Lori, Ilenia Adornato, ... Rosanna Maccari.
35. Chemical constituents from Alismatis Rhizoma and their anti-inflammatory activities in vitro and in vivo
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Shan-shan Liu, Wen-long Sheng, Yun Li, Shan-shan Zhang, ... Mei Zhang.
36. Synthesis, biological evaluation and in silico modelling studies of 1,3,5-trisubstituted pyrazoles carrying benzenesulfonamide as potential anticancer agents and selective cancer-associated hCA IX isoenzyme inhibitors
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Cem Yamali, Halise Inci Gul, Abdulilah Ece, Silvia Bua, ... Claudiu T. Supuran.
37. Design, synthesis, in vitro evaluation, molecular docking and ADME properties studies of hybrid bis-coumarin with thiadiazole as a new inhibitor of Urease
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Munther Alomari, Muhammad Taha, Syahrul Imran, Waqas Jamil, ... Fazal Rahim.
38. Dual-targeting antitumor conjugates derived from platinum(IV) prodrugs and microtubule inhibitor CA-4 significantly exhibited potent ability to overcome cisplatin resistance
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Xiaochao Huang, Meng Wang, Chungu Wang, Weiwei Hu, ... Hengshan Wang.
39. Development of novel chromeno[4,3-c]pyrazol-4(2H)-one derivates containing piperazine as inhibitors of PI3Kα
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Yong Yin, Yang Zhou, Shao Sha, Xun Wu, ... Hai-Liang Zhu.
40. The modulating effect of lipid bilayer/p-coumaric acid interactions on electrical properties of model lipid membranes and human glioblastoma cells
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Monika Naumowicz, Magdalena Kusaczuk, Marcin Andrzej Kruszewski, Miroslav Gál, ... Joanna Kotyńska.
41. Design, synthesis and biological evaluation of theophylline containing variant acetylene derivatives as α-amylase inhibitors
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Radhakrishnam Raju Ruddarraju, Gangarapu Kiran, Adharvana Chari Murugulla, Ravichandar Maroju, ... Nukala Shravya Reddy.
42. New series of fused pyrazolopyridines: Synthesis, molecular modeling, antimicrobial, antiquorum-sensing and antitumor activities
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N.S. El-Gohary, S.S. Hawas, M.T. Gabr, M.I. Shaaban, M.B. El-Ashmawy.
43. Design, synthesis and molecular docking of novel pyrazolo[1,5-a][1,3,5]triazine derivatives as CDK2 inhibitors
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Khulood H. Oudah, Mazin A.A. Najm, Nermin Samir, Rabah A.T. Serya, Khaled A.M Abouzid.
44. Anti-inflammatory flavonoids from root bark of Broussonetia papyrifera in LPS-stimulated RAW264.7 cells
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Hyung Won Ryu, Mi Hyeon Park, Ok-Kyoung Kwon, Doo-Young Kim, ... Sei-Ryang Oh.
45. Variedly connected 1,8-naphthalimide-7-chloroquinoline conjugates: Synthesis, anti-mycobacterial and cytotoxic evaluation
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Shalini, Matt D. Johansen, Laurent Kremer, Vipan Kumar.
46. Tyrosinase inhibitory effects of Vinca major and its secondary metabolites: Enzyme kinetics and in silico inhibition model of the metabolites validated by pharmacophore modelling
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Suat Sari, Burak Barut, Arzu Özel, Didem Şöhretoğlu.
47. Discovery and optimization of 5,7-dihydro-6H-pyrrolo[2,3-d]pyrimidin-6-one derivatives as mTORC1/mTORC2 dual inhibitors
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Tác giả
Shengquan Hu, Zhichang Zhao, Hong Yan.
48. Juniperanol: First total synthesis and evaluation in Type 2 Diabetes disease
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A. Carrër, S. Turban, N. Provost, A. Caliez, ... V. Michelet.
49. Exploring antidiabetic potential of adamantyl-thiosemicarbazones via aldose reductase (ALR2) inhibition
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Muhammad Tariq Shehzad, Abdul Hameed, Mariya al-Rashida, Aqeel Imran, ... Jamshed Iqbal.
50. Design, synthesis, and biological evaluation of novel dual FFA1 (GPR40)/PPARδ agonists as potential anti-diabetic agents
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Zheng Li, Lijun Hu, Xuekun Wang, Zongtao Zhou, ... Luyong Zhang.
51. Effects of Picrasma quassioides and its active constituents on Alzheimer's disease in vitro and in vivo
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Eryan Guo, Yunwei Hu, Tao Du, Huilin Zhu, ... Jian Xu.
52. First example of Azo-Sulfa conjugated chromene moieties: Synthesis, characterization, antimicrobial assessment, docking simulation as potent class I histone deacetylase inhibitors and antitumor agents
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Rawda M. Okasha, Mosa Alsehli, Saleh Ihmaid, Sultan S. Althagfan, ... Tarek H. Afifi.
53. Molecular interaction of manganese based carbon monoxide releasing molecule (MnCORM) with human serum albumin (HSA)
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Pitchavel Vidhyapriya, Dhanaraj Divya, Bala. Manimaran, Natarajan Sakthivel.
54. Anti-cancer activity of the cell membrane-permeable phytic acid prodrug
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Takuya Masunaga, Naoki Murao, Hiroshi Tateishi, Ryoko Koga, ... Mikako Fujita.
55. Design and synthesis of novel pyridazinoquinazoline derivatives as potent VEGFR-2 inhibitors: In vitro and in vivo study
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Marwa G. El-Gazzar, Rania M. El-Hazek, Nashwa H. Zaher, Mona A. El-Ghazaly.
56. New carboxamides bearing benzenesulphonamides: Synthesis, molecular docking and pharmacological properties
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Florence Uchenna Eze, Uchechukwu Chris Okoro, David Izuchukwu Ugwu, Sunday N. Okafor.
57. Novel [1,2,4]triazolo[1,5-a]pyrimidine derivatives as potent antitubulin agents: Design, multicomponent synthesis and antiproliferative activities
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Fang Yang, Liang-Zhentian Yu, Peng-Cheng Diao, Xie-Er Jian, ... Pei-Liang Zhao.
58. Synthesis and biological evaluation of thiazolidine-2,4-dione-pyrazole conjugates as antidiabetic, anti-inflammatory and antioxidant agents
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Garima Bansal, Shamsher Singh, Vikramdeep Monga, Punniyakoti Veeraveedu Thanikachalam, Pooja Chawla.
59. Novel 2-arylthiopropanoyl-CoA inhibitors of α-methylacyl-CoA racemase 1A (AMACR; P504S) as potential anti-prostate cancer agents
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Maksims Yevglevskis, Amit Nathubhai, Katty Wadda, Guat L. Lee, ... Matthew D. Lloyd.
60. Identification of novel small-molecule inhibitors of α-methylacyl-CoA racemase (AMACR; P504S) and structure-activity relationships
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Yoana D. Petrova, Katty Wadda, Amit Nathubhai, Maksims Yevglevskis, ... Matthew D. Lloyd.
61. NO inhibitory diterpenoids as potential anti-inflammatory agents from Euphorbia antiquorum
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Lijun An, Yue Liang, Xueyuan Yang, Huimei Wang, ... Yuanqiang Guo.
62. Synthesis, biological evaluation and molecular docking analysis of novel benzopyrimidinone derivatives as potential anti-tyrosinase agents
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Sarra Chortani, Vijaykumar D. Nimbarte, Mabrouk Horchani, Hichem Ben Jannet, Anis Romdhane.
63. Triazolopyridazine derivatives: Synthesis, cytotoxic evaluation, c-Met kinase activity and molecular docking
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Eman M. Ahmed, Nadia A. Khalil, Azza T. Taher, Rana H. Refaey, Yassin M. Nissan.
64. Design, synthesis, and biological activity of Plastoquinone analogs as a new class of anticancer agents
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Nilüfer Bayrak, Hatice Yıldırım, Mahmut Yıldız, Mohamed O. Radwan, ... Halil I. Ciftci.
65. Immunomodulatory activities of zinc(II)phthalocyanine on the mammalian macrophages through p38 pathway: Potential ex vivo immunomodulatory PDT reagents
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Abdulcelil Yüzer, Furkan Ayaz, Mine Ince.
66. Discovery of 2-ethoxy-4-(methoxymethyl)benzamide derivatives as potent and selective PTP1B inhibitors
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Fangzhou Xie, Yaoyao Liang, Yu Xia, Shuhua Luo, ... Lei Fu.
67. In vitro assessment of 3-alkoxy-5-nitroindazole-derived ethylamines and related compounds as potential antileishmanial drugs
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Álvaro Martín-Montes, Benjamín Aguilera-Venegas, Rosa Mª Morales-Martín, Rubén Martín-Escolano, ... Manuel Sánchez-Moreno.
68. Curcumane C and (±)-curcumane D, an unusual seco-cadinane sesquiterpenoid and a pair of unusual nor-bisabolane enantiomers with significant vasorelaxant activity from Curcuma longa
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Ming-Ming Qiao, Fei Liu, Yu Liu, Li Guo, ... Liang Xiong.
69. Antiprotozoal activities of marine polyether triterpenoids
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Ana R. Díaz-Marrero, Atteneri López-Arencibia, Carlos J. Bethencout-Estrella, Francisco Cen-Pacheco, ... José J. Fernández.
70. Synthesis and investigation of inhibitory activities of imidazole derivatives against the metallo-β-lactamase IMP-1
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Omid Khalili Arjomandi, Mahboubeh Kavoosi, Hadi Adibi.
71. New cytotoxic tricycloalternarenes from fungus Alternaria brassicicola
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Fengli Li, Ying Tang, Weiguang Sun, Jiankun Guan, ... Yonghui Zhang.
72. Synthesis of Mitomycin C and decarbamoylmitomycin C N6 deoxyadenosine-adducts
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Maggie Zheng, Seokjin Hwang, Timothy Snyder, Jake Aquilina, ... Elise Champeil.
73. Design, synthesis and antifungal activity evaluation of isocryptolepine derivatives
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Jun-cai Li, Ren-xuan Wang, Yu Sun, Jia-kai Zhu, ... Xiao-fei Shang.
74. Bioactivity-based analysis and chemical characterization of hypoglycemic and antioxidant components from Artemisia argyi
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Jian-Qi Xiao, Wen-Yuan Liu, Hao-peng Sun, Wei Li, ... Jie Zhang.
75. Rational design of some substituted phenyl azanediyl (bis) methylene phosphonic acid derivatives as potential anticancer agents and imaging probes: Computational inputs, chemical synthesis, radiolabeling, biodistribution and gamma scintigraphy
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Tác giả
Mohammed A. Khedr, Hassan M. Rashed, Hamed Farag, Tamer M. Sakr.
76. Geranylated carbazole alkaloids with potential neuroprotective activities from the stems and leaves of Clausena lansium
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Yan-Ping Liu, Jia-Ming Guo, Xiao-Ping Wang, Yun-Yao Liu, ... Yan-Hui Fu.
77. Optimization study towards more potent thiazolidine-2,4-dione IKK-β modulator: Synthesis, biological evaluation and in silico docking simulation
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Ahmed Elkamhawy, Nam youn Kim, Ahmed H.E. Hassan, Jung-eun Park, ... Eun Joo Roh.
78. Novel inhibitors of leukocyte transendothelial migration
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Tác giả
Tamar Getter, Raanan Margalit, Shirin Kahremany, Laura Levy, ... Arie Gruzman.
79. New triazinoindole bearing thiazole/oxazole analogues: Synthesis, α-amylase inhibitory potential and molecular docking study
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Tác giả
Fazal Rahim, Sundas Tariq, Muhammad Taha, Hayat Ullah, ... Syed Adnan Ali Shah.
80. Targeted 8-hydroxyquinoline fragment based small molecule drug discovery against neglected botulinum neurotoxin type F
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Ritika Chauhan, Vinita Chauhan, Priyanka Sonkar, Manorama Vimal, Ram Kumar Dhaked.
81. Chemical constituents and synergistic anti-gout studies on Eurycoma longifolia and potential mechanisms evaluation based on systemic analysis approach
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Tác giả
Ying Liu, Lantao Lai, Yan Ju, Caihong Liu, Dali Meng.
82. Novel pyridazinone derivatives as butyrylcholinesterase inhibitors
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Tác giả
Yasemin Dundar, Ozge Kuyrukcu, Gokcen Eren, F. Sezer Senol Deniz, ... Ilkay Erdogan Orhan.
83. Discovery of diverse diterpenoid scaffolds from Euphorbia antiquorum and their activity against RANKL-induced osteoclastogenesis
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Zhi-Yong Yin, Yan Dai, Pei Hua, Zhe-Jun Sun, ... Qiong Gu.
84. Umbelliferone derivatives exert neuroprotective effects by inhibiting monoamine oxidase A, self-amyloidβ aggregation, and lipid peroxidation
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Tác giả
Su Hui Seong, Md Yousof Ali, Hyun Ah Jung, Jae Sue Choi.
85. Synthesis and biological evaluation of tetrazole derivatives as TNF-α, IL-6 and COX-2 inhibitors with antimicrobial activity: Computational analysis, molecular modeling study and region-specific cyclization using 2D NMR tools
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Tác giả
Phoebe F. Lamie, Ahmed F. Azmey.
86. 2-Styrylchromone derivatives as potent and selective monoamine oxidase B inhibitors
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Tác giả
Koichi Takao, Saki Endo, Junko Nagai, Hitoshi Kamauchi, ... Yoshiaki Sugita.
87. Design, synthesis, in-vitro evaluation and molecular docking studies of novel indole derivatives as inhibitors of SIRT1 and SIRT2
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Ramu Manjula, Nikhila Gokhale, Sruthi Unni, Prashant Deshmukh, ... Balasundaram Padmanabhan.
88. Discovery, molecular dynamic simulation and biological evaluation of structurally diverse cholinesterase inhibitors with new scaffold through shape-based pharmacophore virtual screening
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Hongyu Yang, Chenxi Du, Qihang Li, Tingkai Chen, ... Haopeng Sun.
89. Synthesis and investigation of polyhydroxylated pyrrolidine derivatives as novel chemotypes showing dual activity as glucosidase and aldose reductase inhibitors
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Lorenzo Guazzelli, Felicia D'Andrea, Stefania Sartini, Francesco Giorgelli, ... Concettina La Motta.
90. Synthesis, structural characterization and in vivo anti-diabetic evaluation of some new sulfonylurea derivatives in normal and silicate coated nanoparticle forms as anti-hyperglycemic agents
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Farid M. Sroor, Samir Y. Abbas, Wahid M. Basyouni, Khairy A.M. El-Bayouki, ... Ahmed A. Haroun.
91. Arylpropionic acid-derived NSAIDs: New insights on derivatization, anticancer activity and potential mechanism of action
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Ahmed M. Gouda, Eman A. Beshr, Faisal A. Almalki, Hadeel H. Halawah, ... Malak M. AlMatrafi.
92. Disulfide bridge as a linker in nucleic acids’ bioconjugation. Part I: An overview of synthetic strategies
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Anna R. Stasińska, Piotr Putaj, Marcin K. Chmielewski.
93. The role of long noncoding RNA in major human disease
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Tác giả
Xiaoli Zhang, Ruiyun Hong, Weiqiang Chen, Minwen Xu, Liefeng Wang.
94. Promising antibacterial agents against multidrug resistant Staphylococcus aureus
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Tác giả
Srikanth Gatadi, Y.V. Madhavi, Sidharth Chopra, Srinivas Nanduri.
95. Recent advances in the synthetic and medicinal perspective of quinolones: A review
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Tác giả
Prashant Dhiman, Nidhi Arora, Punniyakoti Veeraveedu Thanikachalam, Vikramdeep Monga.
96. Identification of potential inflammatory inhibitors from Aster tataricus
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Tác giả
Xiang Dong Su, Hyun-Jae Jang, Hong Xu Li, Young Ho Kim, Seo Young Yang.
97. New pyrimidine-benzoxazole/benzimidazole hybrids: Synthesis, antioxidant, cytotoxic activity, in vitro cyclooxygenase and phospholipase A2-V inhibition
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Mohamed A. Abdelgawad, Rania B. Bakr, Waqas Ahmad, Mohammad M. Al-Sanea, Heba A.H. Elshemy.
98. Design, synthesis and biological evaluation of some tetrazole acetamide derivatives as novel non-carboxylic PTP1B inhibitors
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Neelesh Maheshwari, Chandrabose Karthikeyan, Shraddha V. Bhadada, Amit K. Verma, ... Piyush Trivedi.
99. A novel adaptive fluorescent probe for cell labelling
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Anca G. Coman, Anca Paun, Codruta C. Popescu, Niculina D. Hădade, ... Mihaela Matache.
100. Discovery of a series of selective and cell permeable beta-secretase (BACE1) inhibitors by fragment linking with the assistance of STD-NMR
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Wei-Shuo Fang, De-yang Sun, Shuang Yang, Chen Cheng, ... Yinghong Wang.
