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Bioorganic Chemistry
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Volume 89, August 2019, Hidden issue
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1. Editorial Board
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2. Issue TOC
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3. Follow on-based optimization of the biphenyl-DAPYs as HIV-1 nonnucleoside reverse transcriptase inhibitors against the wild-type and mutant strains
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Yali Sang, Sheng Han, Shuwen Han, Christophe Pannecouque, ... Fener Chen.
4. Synthesis, molecular modeling and biological evaluation of new pyrazolo[3,4-b]pyridine analogs as potential antimicrobial, antiquorum-sensing and anticancer agents
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N.S. El-Gohary, M.T. Gabr, M.I. Shaaban.
5. Design and synthesis of new benzoxazole/benzothiazole-phthalimide hybrids as antitumor-apoptotic agents
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Tác giả
John N. Philoppes, Phoebe F. Lamie.
6. An efficient one-pot synthesis of polyphenolic amino acids and evaluation of their radical-scavenging activity
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Luís S. Monteiro, Fátima Paiva-Martins, Sandra Oliveira, Inês Machado, Marlene Costa.
7. Syntesis of thio- and seleno-acetamides bearing benzenesulfonamide as potent inhibitors of human carbonic anhydrase II and XII
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Damiano Tanini, Antonella Capperucci, Martina Scopelliti, Andrea Milaneschi, ... Claudiu T. Supuran.
8. Synthesis and in vitro anticancer evaluation of some fused indazoles, quinazolines and quinolines as potential EGFR inhibitors
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Esraa A. Abdelsalam, Wafaa A. Zaghary, Kamilia M. Amin, Nageh A. Abou Taleb, ... Sherif F. Hammad.
9. Synthesis, biological evaluation and in silico studies of novel N-substituted phthalazine sulfonamide compounds as potent carbonic anhydrase and acetylcholinesterase inhibitors
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Cüneyt Türkeş, Mustafa Arslan, Yeliz Demir, Liridon Çoçaj, ... Şükrü Beydemir.
10. Catechol thioethers with physiologically active fragments: Electrochemistry, antioxidant and cryoprotective activities
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Ivan V. Smolyaninov, Olga V. Pitikova, Eugenia O. Korchagina, Andrey I. Poddel'sky, ... Nadezhda T. Berberova.
11. Antitrypanosomal activity and effect in plasma membrane permeability of (−)-bornyl p-coumarate isolated from Piper cernuum (Piperaceae)
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Thiago R. Morais, Thais A. Costa-Silva, Daiane D. Ferreira, Bianca J. Novais, ... João Henrique G. Lago.
12. Evaluation of the antitrypanosoma activity and SAR study of novel LINS03 derivatives
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Marina T. Varela, Thais A. Costa-Silva, João Henrique G. Lago, Andre G. Tempone, João Paulo S. Fernandes.
13. Synthesis, biological evaluation and molecular docking studies of novel 3,5-disubstituted 2,4-thiazolidinediones derivatives
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Alok Ranjan Srivastava, Rohit Bhatia, Pooja Chawla.
14. Tetrahydro-1H,5H-pyrazolo[1,2-a]pyrazole-1-carboxylates as inhibitors of Plasmodium falciparum dihydroorotate dehydrogenase
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Nika Strašek, Lara Lavrenčič, Andraž Oštrek, Dejan Slapšak, ... Jurij Svete.
15. Targeting malaria and leishmaniasis: Synthesis and pharmacological evaluation of novel pyrazole-1,3,4-oxadiazole hybrids. Part II
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Garima Verma, Mohemmed Faraz Khan, Lalit Mohan Nainwal, Mohd Ishaq, ... Mohammad Shaquiquzzaman.
16. 3D-QSAR pharmacophore modelling, virtual screening and docking studies for lead discovery of a novel scaffold for VEGFR 2 inhibitors: Design, synthesis and biological evaluation
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Mahitab K. Sobhy, Samar Mowafy, Deena S. Lasheen, Nahla A. Farag, Khaled A.M. Abouzid.
17. Molecular docking and experimental investigation of new indole derivative cyclooxygenase inhibitor to probe its binding mechanism with bovine serum albumin
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Tanveer A. Wani, Ahmed H. Bakheit, Seema Zargar, Mashooq A. Bhat, Abdulrahman A. Al-Majed.
18. Design and synthesis of dye-conjugated hepsin inhibitors
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Kyul Kim, Hongmok Kwon, Doyoung Choi, Taehyeong Lim, ... Youngjoo Byun.
19. EGFR inhibitors and apoptotic inducers: Design, synthesis, anticancer activity and docking studies of novel xanthine derivatives carrying chalcone moiety as hybrid molecules
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Hesham A. Abou-Zied, Bahaa G.M. Youssif, Mamdouh F.A. Mohamed, Alaa M. Hayallah, Mohamed Abdel-Aziz.
20. Antitrypanosomal activity of isololiolide isolated from the marine hydroid Macrorhynchia philippina (Cnidaria, Hydrozoa)
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Marta L. Lima, Maiara M. Romanelli, Samanta E.T. Borborema, Deidre M. Johns, ... Andre G. Tempone.
21. Synthesis, thymidine phosphorylase, angiogenic inhibition and molecular docking study of isoquinoline derivatives
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Khalid Zaman, Fazal Rahim, Muhammad Taha, Abdul Wadood, ... Ashfaq Ahmed.
22. Structure-based design and synthesis of new 4-methylcoumarin-based lignans as pro-inflammatory cytokines (TNF-α, IL-6 and IL-1β) inhibitors
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S. Santhosh Kumar, Ahil Sajeli Begum, Kirti Hira, Sarfaraj Niazi, ... Yoshinori Fujimoto.
23. Biosynthesized silver nanoparticles for inhibition of antibacterial resistance and biofilm formation of methicillin-resistant coagulase negative Staphylococci
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Govindan Rajivgandhi, Muthuchamy Maruthupandy, Thillaichidambaram Muneeswaran, Muthusamy Anand, ... Wen-Jun Li.
24. Synthesis of 1-benzyl-1H-benzimidazoles as galectin-1 mediated anticancer agents
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Nerella Sridhar Goud, S. Mahammad Ghouse, Jatoth Vishnu, D. Komal, ... Mallika Alvala.
25. Design, synthesis, in vivo, and in silico evaluation of new coumarin-1,2,4-oxadiazole hybrids as anticonvulsant agents
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Maryam Mohammadi-Khanaposhtani, Nematollah Ahangar, Sepideh Sobhani, Patrick Honarchian Masihi, ... Tahmineh Akbarzadeh.
26. Pharmacological investigation of quinoxaline-bisthiazoles as multitarget-directed ligands for the treatment of Alzheimer’s disease
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Sneha R. Sagar, Devendra Pratap Singh, Rajesh D. Das, Nirupa B. Panchal, ... Kamala K. Vasu.
27. Design, synthesis and biological activity of novel tacrine-isatin Schiff base hybrid derivatives
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E. Riazimontazer, H. Sadeghpour, H. Nadri, A. Sakhteman, ... N. Edraki.
28. Synthesis, molecular properties, anti-inflammatory and anticancer activities of novel 3-hydroxyflavone derivatives
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Mansour Znati, Claire Bordes, Valérian Forquet, Pierre Lantéri, ... Jalloul Bouajila.
29. Strophasterols E and F: Rearranged ergostane-type sterols from Pleurotus eryngii
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Takashi Kikuchi, Maya Isobe, Sawako Uno, Yasuko In, ... Takeshi Yamada.
30. Phototoxicity of 7-oxycoumarins with keratinocytes in culture
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Christophe Guillon, Yi-Hua Jan, Diane E. Heck, Thomas M. Mariano, ... Ned D. Heindel.
31. Design, synthesis and molecular modeling studies of new series of s-triazine derivatives as antimicrobial agents against multi-drug resistant clinical isolates
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Nesreen Saied Haiba, Hosam H. Khalil, Mohamed Abdel Moniem, Marwa H. El-Wakil, ... Sherine Nabil Khattab.
32. Synthesis and biological evaluation of aryl phosphoramidate prodrugs of fosfoxacin and its derivatives
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Mathilde Munier, Denis Tritsch, Didier Lièvremont, Michel Rohmer, Catherine Grosdemange-Billiard.
33. Identification of 2(1H)-pyrimidinones as potential EGFR T790M inhibitors for the treatment of gefitinib-resistant non-small cell lung cancer
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Jianping Huang, Jiaxin Huang, Ning Wang, Luhong Wang, ... Xiaodong Ma.
34. Synthesis and biological evaluation of bromophenol derivatives with cyclopropyl moiety: Ring opening of cyclopropane with monoester
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Murat Boztas, Parham Taslimi, Mirali Akbar Yavari, Ilhami Gulcin, ... Abdullah Menzek.
35. A bright blue fluorescent dextran for two-photon in vivo imaging of blood vessels
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Seo Hyeon Lee, Young Ho Choe, Rae Hyung Kang, Yu Rim Kim, ... Dokyoung Kim.
36. Design and development of 1,3,4-oxadiazole derivatives as potential inhibitors of acetylcholinesterase to ameliorate scopolamine-induced cognitive dysfunctions
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Puja Mishra, Piyoosh Sharma, Prabhash Nath Tripathi, Sukesh Kumar Gupta, ... Sushant Kumar Shrivastava.
37. Design, synthesis and biological evaluation of pyrazolopyrimidinone based potent and selective PDE5 inhibitors for treatment of erectile dysfunction
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G. Lakshma Reddy, Mohd. Ishaq Dar, Abhinandan D. Hudwekar, Priya Mahajan, ... Sanghapal D. Sawant.
38. Cytotoxic diterpenoids as potential anticancer agents from the twigs of Casearia kurzii
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Feng Liu, Qi Zhang, Xueyuan Yang, Yaru Xi, ... Yuanqiang Guo.
39. Bridged bicyclic 2,3-dioxabicyclo[3.3.1]nonanes as antiplasmodial agents: Synthesis, structure-activity relationships and studies on their biomimetic reaction with Fe(II)
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Sarah D'Alessandro, Gloria Alfano, Luisa Di Cerbo, Simone Brogi, ... Stefania Butini.
40. Radical scavenging and anti-inflammatory activities of (hetero)arylethenesulfonyl fluorides: Synthesis and structure-activity relationship (SAR) and QSAR studies
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Ying Jiang, K.P. Rakesh, Njud S. Alharbi, H.K. Vivek, ... Hua-Li Qin.
41. Design, synthesis, modeling studies and biological screening of novel pyrazole derivatives as potential analgesic and anti-inflammatory agents
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Azza T. Taher, Marwa T. Mostafa Sarg, Nermeen R. El-Sayed Ali, Noha Hilmy Elnagdi.
42. Synthesis, in vitro urease inhibitory potential and molecular docking study of Benzimidazole analogues
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Khalid Zaman, Fazal Rahim, Muhammad Taha, Hayat Ullah, ... Mohammed Gollapalli.
43. Novel chromanone-dithiocarbamate hybrids as multifunctional AChE inhibitors with β-amyloid anti-aggregation properties for the treatment of Alzheimer’s disease
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Neng Jiang, Jiaoli Ding, Jing Liu, Xiaona Sun, ... Sai-Sai Xie.
44. Discovery of novel (+)-Usnic acid derivatives as potential anti-leukemia agents with pan-Pim kinases inhibitory activity
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Shuxiang Wang, Jie Zang, Min Huang, Lihong Guan, ... Linxiang Zhao.
45. An NIR emitting styryl dye with large Stokes shift to enable co-staining study on zebrafish neuromast hair cells
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Lucas McDonald, Dipendra Dahal, Michael Konopka, Qin Liu, Yi Pang.
46. Design, synthesis and anticervical cancer activity of new benzofuran–pyrazol-hydrazono- thiazolidin-4-one hybrids as potential EGFR inhibitors and apoptosis inducing agents
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Hebat-Allah S. Abbas, Somaia S. Abd El-Karim.
47. Structural basis of the inhibition of GH1 β-glucosidases by multivalent pyrrolidine iminosugars
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Macarena Martínez-Bailén, Elena Jiménez-Ortega, Ana T. Carmona, Inmaculada Robina, ... Antonio J. Moreno-Vargas.
48. Potent inhibition of acetylcholinesterase by sargachromanol I from Sargassum siliquastrum and by selected natural compounds
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Jae Pil Lee, Myung-Gyun Kang, Joon Yeop Lee, Jong Min Oh, ... Hoon Kim.
49. N-aryl-N’-ureido-O-sulfamates: Potent and selective inhibitors of the human Carbonic Anhydrase VII isoform with neuropathic pain relieving properties
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Murat Bozdag, Giulio Poli, Andrea Angeli, Elena Lucarini, ... Claudiu T. Supuran.
50. Discovery of pyrazolopyrimidine derivatives as potent BTK inhibitors with effective anticancer activity in MCL
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Fansheng Ran, Yang Liu, Meixia Liu, Daoguang Zhang, ... Guisen Zhao.
51. Novel imidazo[2,1-b][1,3,4]thiadiazole (ITD) hybrid compounds: Design, synthesis, efficient antibacterial activity and antioxidant effects
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Ebru Taflan, Hacer Bayrak, Mehtap Er, Şengül Alpay Karaoğlu, Arif Bozdeveci.
52. Recent advancement in the discovery and development of COX-2 inhibitors: Insight into biological activities and SAR studies (2008–2019)
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Vrinda Sharma, Parth Bhatia, Ozair Alam, Mohd. Javed Naim, ... Mukund Jha.
53. Medicinal chemistry of indole derivatives: Current to future therapeutic prospectives
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Archana Kumari, Rajesh K. Singh.
54. Rational design, synthesis and biological evaluation of ubiquinone derivatives as IDO1 inhibitors
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Yuyang Ding, Fei Tang, Xiaoqian Xue, Jinfeng Luo, ... Jiancun Zhang.
55. Design, synthesis and evaluation of phenylfuroxan nitric oxide-donor phenols as potential anti-diabetic agents
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Yun-Dong Xie, Li-Hua Shao, Qiu-Tang Wang, Yue Bai, ... Xiao-Li Bian.
56. Exploring the competence stimulating peptide (CSP) N-terminal requirements for effective ComD receptor activation in group1 Streptococcus pneumoniae
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Yifang Yang, Yftah Tal-Gan.
