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Bioorganic Chemistry
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Volume 85, Pages 1-600 (April 2019), Hidden issue
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1. Editorial Board
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2. Issue TOC
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3. Syntheses and evaluation of new Quinoline derivatives for inhibition of hnRNP K in regulating oncogene c-myc transcription
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Bing Shu, Ping Zeng, Shuangshuang Kang, Peng-Hui Li, ... Ding Li.
4. Ursolic and oleanolic acid derivatives with cholinesterase inhibiting potential
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Anne Loesche, Alexander Köwitsch, Susana D. Lucas, Zayan Al-Halabi, ... René Csuk.
5. Synthesis of benzothiazole derivatives as a potent α-glucosidase inhibitor
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Mohammed Gollapalli, Muhammad Taha, Muhammad Tariq Javid, Noor Barak Almandil, ... Yasser A. Bamarouf.
6. Synthesis, molecular properties prediction and biological evaluation of indole-vinyl sulfone derivatives as novel tubulin polymerization inhibitors targeting the colchicine binding site
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Wenlong Li, Honghao Sun, Feijie Xu, Wen Shuai, ... Jinyi Xu.
7. The monoamine oxidase inhibition properties of C6-mono- and N3/C6-disubstituted derivatives of 4(3H)-quinazolinone
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Malikotsi A. Qhobosheane, Lesetja J. Legoabe, Anél Petzer, Jacobus P. Petzer.
8. Synthesis and biological activity of a potent optically pure autoinducer-2 quorum sensing agonist
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Osvaldo S. Ascenso, Inês M. Torcato, Ana Sofia Miguel, João C. Marques, ... Christopher D. Maycock.
9. Biphenyl-3-oxo-1,2,4-triazine linked piperazine derivatives as potential cholinesterase inhibitors with anti-oxidant property to improve the learning and memory
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Prabhash Nath Tripathi, Pavan Srivastava, Piyoosh Sharma, Manish Kumar Tripathi, ... Sushant K. Shrivastava.
10. In vitro and in silico evaluation of new thiazole compounds as monoamine oxidase inhibitors
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Begüm Nurpelin Sağlık, Betül Kaya Çavuşoğlu, Derya Osmaniye, Serkan Levent, ... Yusuf Öztürk.
11. Synthesis of novel quinoline-based thiadiazole, evaluation of their antileishmanial potential and molecular docking studies
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Noor Barak Almandil, Muhammad Taha, Fazal Rahim, Abdul Wadood, ... Mohammed Gollapalli.
12. Expansion of the scaffold diversity for the development of highly selective butyrylcholinesterase (BChE) inhibitors: Discovery of new hits through the pharmacophore model generation, virtual screening and molecular dynamics simulation
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Xin Lu, Hongyu Yang, Qihang Li, Yao Chen, ... Haopeng Sun.
13. The first synthesis, carbonic anhydrase inhibition and anticholinergic activities of some bromophenol derivatives with S including natural products
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Cetin Bayrak, Parham Taslimi, Halide Sedef Karaman, Ilhami Gulcin, Abdullah Menzek.
14. 3, 9-di-O-substituted coumestrols incorporating basic amine side chains act as novel apoptosis inducers with improved pharmacological selectivity
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Guoshun Luo, Zhengpu Tang, Xinyu Li, Qiangqiang Hou, ... Hua Xiang.
15. Cloning, overexpression and characterization of a thermostable β-xylosidase from Thermotoga petrophila and cooperated transformation of ginsenoside extract to ginsenoside 20(S)-Rg3 with a β-glucosidase
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Shanshan Zhang, Jingcong Xie, Linguo Zhao, Jianjun Pei, ... Zhenzhong Wang.
16. Identification of a pyrimidinetrione derivative as the potent DprE1 inhibitor by structure-based virtual ligand screening
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Ya Gao, Jinshan Xie, Ruotian Tang, Kaiyin Yang, ... Hua Li.
17. Mitochondria-targeted triphenylphosphonium conjugated glycyrrhetinic acid derivatives as potent anticancer drugs
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Le Jin, Lumei Dai, Min Ji, Hengshan Wang.
18. Synthesis and biological evaluation of novel tris-chalcones as potent carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase and α-glycosidase inhibitors
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Serdar Burmaoglu, Ali Osman Yilmaz, M. Fatih Polat, Rüya Kaya, ... Oztekin Algul.
19. Synthesis of novel benzenesulfonamide bearing 1,2,3-triazole linked hydroxy-trifluoromethylpyrazolines and hydrazones as selective carbonic anhydrase isoforms IX and XII inhibitors
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Vikas Sharma, Rajiv Kumar, Silvia Bua, Claudiu T. Supuran, Pawan K. Sharma.
20. Identification of 1,2,4-triazoles as new thymidine phosphorylase inhibitors: Future anti-tumor drugs
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Sohail Anjum Shahzad, Muhammad Yar, Zulfiqar Ali Khan, Lubna Shahzadi, ... Marek Bajda
21. Docking- and pharmacophore-based virtual screening for the identification of novel Mycobacterium tuberculosis protein tyrosine phosphatase B (MptpB) inhibitor with a thiobarbiturate scaffold
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Dongfeng Zhang, Yun Lin, Xi Chen, Wenting Zhao, ... Yu Lu.
22. Exploring the antimalarial potential of the methoxy-thiazinoquinone scaffold: Identification of a new lead candidate
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Concetta Imperatore, Marco Persico, Maria Senese, Anna Aiello, ... Marialuisa Menna.
23. Synthesis, anticancer effect and molecular modeling of new thiazolylpyrazolyl coumarin derivatives targeting VEGFR-2 kinase and inducing cell cycle arrest and apoptosis
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Tahia K. Mohamed, Rasha Z. Batran, Samia A. Elseginy, Mamdouh M. Ali, Abeer E. Mahmoud.
24. Lanceoleins A–G, hydroxychalcones, from the flowers of Coreopsis lanceolata and their chemopreventive effects against human colon cancer cells
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Hyoung-Geun Kim, Hyun-Ji Oh, Jung-Hwan Ko, Hae Seong Song, ... Nam-In Baek.
25. Targeting microbial resistance: Synthesis, antibacterial evaluation, DNA binding and modeling study of new chalcone-based dithiocarbamate derivatives
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Marwa Ayman, Shahenda M. El-Messery, Elsayed E. Habib, Sara T. Al-Rashood, ... Ghada S. Hassan.
26. Design and synthesis of new phthalazine-based derivatives as potential EGFR inhibitors for the treatment of hepatocellular carcinoma
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Ahmed T.A. Boraei, Hanaa K. Ashour, El Sayed H. El Tamany, Nahla Abdelmoaty, ... Mohamed S. Gomaa.
27. Synthesis and biological evaluation of some novel thiobenzimidazole derivatives as anti-renal cancer agents through inhibition of c-MET kinase
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Hany S. Ibrahim, Mohamed E. Albakri, Walaa R. Mahmoud, Heba Abdelrasheed Allam, ... Hatem A. Abdel-Aziz.
28. O-linked melatonin dimers as bivalent ligands targeting dimeric melatonin receptors
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Angeliki Karamitri, Mirna S. Sadek, Anne-Sophie Journé, Florence Gbahou, ... Darius P. Zlotos.
29. Orobanone analogues from acid-promoted aromatization rearrangement of curcumol inhibit hypoxia-inducible factor-1 (HIF-1) in cell-based reporter assays
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Yue-qing Li, Guang-zhe Li, Yi Dong, Xu Ma, ... Wei-jie Zhao.
30. The mechanism of interactions between flavan-3-ols against a-glucosidase and their in vivo antihyperglycemic effects
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Ling-Ling Zhang, Lin Han, Shi-Yi Yang, Xue-Mei Meng, ... Min Wang.
31. Design, synthesis, biological evaluation and molecular modelling studies of indole glyoxylamides as a new class of potential pancreatic lipase inhibitors
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S.N.C. Sridhar, Saksham Palawat, Atish T. Paul.
32. Studies on lysozyme modifications induced by substituted p-benzoquinones
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Jisook Kim, Charles A. Thomas, Jacob M. Ewald, Neethu M. Kurien, ... Titus V. Albu.
33. Design, synthesis, molecular docking and biological activity evaluation of some novel indole derivatives as potent anticancer active agents and apoptosis inducers
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Ahmed M. Sh. El-Sharief, Yousry A. Ammar, Amany Belal, Marwa A.M. Sh. El-Sharief, ... Ahmed Ragab.
34. Synthesis of 1-(α-aminoalkyl)-2-naphthol and α-aminonitrile derivatives with molybdenum Schiff base complex covalently bonded on silica-coated magnetic nanoparticles and DNA interaction study of one type of derivatives using computational and spectroscopi
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Jamshid Rakhtshah, Behrouz Shaabani, Sadegh Salehzadeh, Neda Hosseinpour Moghadam.
35. Synthesis, characterization, antioxidant power and acute toxicity of some new azo-benzamide and azo-imidazolone derivatives with in vivo and in vitro antimicrobial evaluation
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Mohammed Kareem Samad, Farouq Emam Hawaiz.
36. Novel hybrids of podophyllotoxin and formononetin inhibit the growth, migration and invasion of lung cancer cells
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Chengli Yang, Qiongli Xie, Xian Zeng, Nengyin Tao, ... Lei Zhang.
37. Novel lawsone-containing ruthenium(II) complexes: Synthesis, characterization and anticancer activity on 2D and 3D spheroid models of prostate cancer cells
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Rone Aparecido De Grandis, Patrick Wellington da Silva dos Santos, Katia Mara de Oliveira, Ana Rita Tomazela Machado, ... Fernando Rogério Pavan.
38. Click chemistry based multicomponent approach in the synthesis of spirochromenocarbazole tethered 1,2,3-triazoles as potential anticancer agents
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Pramod V. Chavan, Uday V. Desai, Prakash P. Wadgaonkar, Savita R Tapase, ... Dhiman Sarkar.
39. Anti-enteroviral activity of new MDL-860 analogues: Synthesis, in vitro/in vivo studies and QSAR analysis
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Ivanka Nikolova, Ivaylo Slavchev, Martin Ravutsov, Miroslav Dangalov, ... Georgi M. Dobrikov.
40. Absolute configuration and anti-cancer effect of prenylated flavonoids and flavonostilbenes from Sophora pachycarpa: Possible involvement of Wnt signaling pathway
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Motahare Boozari, Samad Nejad Ebrahimi, Saba Soltani, Zahra Tayarani-Najaran, ... Mehrdad Iranshahi.
41. Cell penetrable, clickable and tagless activity-based probe of human cathepsin L
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Dibyendu Dana, Jeremy Garcia, Ashif I. Bhuiyan, Pratikkumar Rathod, ... Sanjai K. Pathak.
42. Design, synthesis and biological study of hybrid drug candidates of nitric oxide releasing cucurbitacin-inspired estrone analogs for treatment of hepatocellular carcinoma
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Mahrous A. Abou-Salim, Mohamed A. Shaaban, Mohammed K. Abd El Hameid, Yaseen A.M.M. Elshaier, Fathi Halaweish.
43. Design, synthesis and evaluation of d-amino acid-containing peptidomimetics targeting the polo-box domain of polo-like kinase 1
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Zhiyan Li, Zhenguo Zhang, Yanhong Chen, Shijun Tang, ... Cheng Jiang.
44. Pyrazoles containing thiophene, thienopyrimidine and thienotriazolopyrimidine as COX-2 selective inhibitors: Design, synthesis, in vivo anti-inflammatory activity, docking and in silico chemo-informatic studies
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Mai S. El-Shoukrofy, Heba A. Abd El Razik, Omaima M. AboulWafa, Aida E. Bayad, Ibrahim M. El-Ashmawy.
45. Cytotoxic clerodane diterpenoids from the leaves of Casearia kurzii
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Jun Ma, Xueyuan Yang, Qi Zhang, Xuke Zhang, ... Yuanqiang Guo.
46. Indole derivatives as multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity of indole hydrazones
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Monica Demurtas, Anna Baldisserotto, Ilaria Lampronti, Davide Moi, ... Valentina Onnis.
47. Novel aryl carboximidamide and 3-aryl-1,2,4-oxadiazole analogues of naproxen as dual selective COX-2/15-LOX inhibitors: Design, synthesis and docking studies
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Bahaa G.M. Youssif, Mamdouh F.A. Mohamed, Mohammad M. Al-Sanea, Amr H. Moustafa, ... Hesham A.M. Gomaa.
48. Design, synthesis, and DNA interaction studies of furo-imidazo[3.3.3]propellane derivatives: Potential anticancer agents
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Alaa A. Hassan, Ashraf A. Aly, Nasr K. Mohamed, Kamal M. El Shaieb, ... Tamer S. Kaoud.
49. Bio-guided search of active indole alkaloids from Tabernaemontana catharinensis: Antitumour activity, toxicity in silico and molecular modelling studies
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Pauline Fagundes Rosales, Flavio Ferreira Marinho, Adriana Gower, Marilda Chiarello, ... Sidnei Moura.
50. Piperazine-azole-fluoroquinolone hybrids: Conventional and microwave irradiated synthesis, biological activity screening and molecular docking studies
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Arif Mermer, Ozlem Faiz, Ahmet Demirbas, Neslihan Demirbas, ... Sivakumar Arumugam.
51. Wedtrilosides A and B, two new diterpenoid glycosides from the leaves of Wedelia trilobata (L.) Hitchc. with α-amylase and α-glucosidase inhibitory activities
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Nguyen Thi Luyen, Pham Thanh Binh, Pham Thi Tham, Ta Manh Hung, ... Nguyen Phuong Thao.
52. A molecular hybrid producing simultaneously singlet oxygen and nitric oxide by single photon excitation with green light
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Cristina Parisi, Mariacristina Failla, Aurore Fraix, Antonio Rescifina, ... Salvatore Sortino.
53. Radicicol rescues yeast cell death triggered by expression of human α-synuclein and its A53T mutant, but not by human βA4 peptide and proapoptotic protein bax
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Asma Derf, Shilpa A. Verekar, Shreyans K. Jain, Sunil K. Deshmukh, ... Bhabatosh Chaudhuri.
54. Synthesis, antioxidant and Aβ anti-aggregation properties of new ferulic, caffeic and lipoic acid derivatives obtained by the Ugi four-component reaction
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Mohamed Benchekroun, Irene Pachón-Angona, Vincent Luzet, Helene Martin, ... Lhassane Ismaili.
55. Innovative nano-carriers in anticancer drug delivery-a comprehensive review
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Peng Dong, K.P. Rakesh, H.M. Manukumar, Yasser Hussein Eissa Mohammed, ... Hua-Li Qin.
56. Bioactive cytosporone derivatives isolated from the mangrove-derived fungus Dothiorella sp. ML002
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Cai-Juan Zheng, Guo-Lei Huang, Hai-Xia Liao, Rong-Qing Mei, ... Qing-Ying Zhang.
57. Discovery of atorvastatin as a tetramer stabilizer of nuclear receptor RXRα through structure-based virtual screening
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Xin Wang, Shuyi Chong, Huiyun Lin, Zhiqiang Yan, ... Ying Su.
58. Chiral resolution and neuroprotective activities of enantiomeric dihydrobenzofuran neolignans from the fruit of Crataegus pinnatifida
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Rui Guo, Tian-Ming Lv, Feng-Ying Han, Bin Lin, ... Shao-Jiang Song.
